| Year | Detail |
| 1941 |
Nihon Eisai Co. Ltd. is established in Saitama, eastern Japan. |
| 1944 |
Sakuragaoka Laboratory Co. Ltd. and Nihon Eisai Co. Ltd. merge under the name Nihon Eisai Co. Ltd. |
| 1950 |
Launched cardiotonic Neophyllin in Japan. |
| 1952 |
Nihon Eisai Co. Ltd. launches high-dosage vitamin B1 and B2 product Chocola BB Tablets in Japan. |
| 1955 |
The company changes its name from Nihon Eisai Co. Ltd. to Eisai Co. Ltd. |
| 1961 |
Eisai opens its Taipei Office. |
| 1969 |
Youda Co. Ltd. is established as a pharmaceutical imports subsidiary in Taiwan. |
| 1970 |
PT Eisai Indonesia is established. |
| 1971 |
Toyoji opens the Naito Museum of Pharmaceutical Science and Industry. |
| 1974 |
Eisai (Malaysia) Sdn. Bhd. and Hi-Eisai Pharmaceutical Inc. are established as pharmaceutical sales subsidiaries in Malaysia and the Philippines, respectively. |
| 1977 |
Launched Naturally derived vitamin E product Juvelux. |
| 1981 |
Eisai U.S.A. Inc. is established. |
| 1982 |
The Tsukuba Research Laboratories open in Ibaraki, eastern Japan. |
| 1989 |
Eisai Machinery GmbH is established in Germany. |
| 1995 |
Eisai Inc. is established as a pharmaceutical sales subsidiary in New Jersey, the U.S. |
| 1998 |
Aricept is launched in France. |
| 2004 |
Eisai Europe Ltd. is established. |
| 2008 |
Eisai acquires MGI Pharma Inc. |
| 2018 |
Eisai agrees upon a strategic collaboration for Lenvima with Merck & Co. Inc. and Kenilworth. |
| 2020 |
Unlimit Health Limited is established in Shanghai, China. |
| 2022 |
Eisai Pharmaceuticals Africa (Pty) Ltd is established. |
| 2023 |
LEQEMBI is launched in Japan. |